Meperidine

Meperidine

  • Opioid analgesic
  • Strong opioid agonist
  • Activates opioid receptors

  •  Inhibits pain transmission

  •  Generalized CNS depression

  •  Moderate-severe pain

  •  Analgesia during labor

  •  Preoperative sedation

  •  Lacks antitussive activity

  •  Confusion

  •  Sedation

  •  Constipation

  •  N, V

  •  Dependence

  •  Toxic metabolite CNS excitation, convulsions, tremors

  •  AVOID MAOI >>> Potentially fatal

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